SR 8278 |CAS:1254944-66-5 Probechem Biochemicals

Chemical Structure : SR 8278

CAS No.: 1254944-66-5

SR 8278 (SR8278)

Catalog No.: PC-62691Not For Human Use, Lab Use Only.

SR 8278 is the first synthetic antagonist of the nuclear heme receptor Rev-ErbA, inhibits the REV-ERBα transcriptional repression activity with EC50 of 0.47 uM in HEK293 cells..

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25 mg	$328	In stock
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Biological Activity

SR 8278 is the first synthetic antagonist of the nuclear heme receptor Rev-ErbA, inhibits the REV-ERBα transcriptional repression activity with EC50 of 0.47 uM in HEK293 cells.

Physicochemical Properties

M.Wt	361.48
Formula	C18H19NO3S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1,2,3,4-Tetrahydro-2-[[5-(methylthio)-2-thienyl]carbonyl]-3-isoquinolinecarboxylic acid ethyl ester

References

1. Kojetin D, et al. ACS Chem Biol. 2011 Feb 18;6(2):131-4.

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SR 8278 (SR8278)

Biological Activity

Physicochemical Properties

References

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