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SRPIN803

Chemical Structure : SRPIN803

CAS No.: 380572-02-1

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SRPIN803 (SRPIN-803)

Catalog No.: PC-60568Not For Human Use, Lab Use Only.

SRPIN803 is a novel small molecule dual inhibitor of SRPK1 and CK2 with IC50 of 2.4 uM and 0.2 uM, respectively, does not inhibit SRPK2.

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5 mg $148 In stock
10 mg $228 In stock
25 mg $378 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

SRPIN803 is a novel small molecule dual inhibitor of SRPK1 and CK2 with IC50 of 2.4 uM and 0.2 uM, respectively, does not inhibit SRPK2.
SRPIN803 prevents VEGF production more effectively than SRPIN340, topical administration of SRPIN803 suppresses intraocular neovascularization in mouse model.

Physicochemical Properties

M.Wt 370.306
Formula C14H9F3N4O3S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

5,6-Dihydro-6-[(4-hydroxy-3-methoxyphenyl)methylene]-5-imino-2-(trifluoromethyl)-7H-1,3,4-thiadiazolo[3,2-a]pyrimidin-7-one

References

1. Morooka S, et al. Mol Pharmacol. 2015 Aug;88(2):316-25.

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