Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-GPCR-Adenosine Receptor-ST1535
ST1535

Chemical Structure : ST1535

CAS No.: 496955-42-1

ST1535 (ST 1535;ST-1535)

Catalog No.: PC-70072Not For Human Use, Lab Use Only.

ST1535 is a potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.

Packing Price Stock Quantity
10 mg $188 In stock
25 mg $298 In stock
50 mg $488 In stock
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

ST1535 is a potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
ST1535 displays 10, 58 and >160-fold selectivity over A1, A2B and A3 receptors, respectively.
ST1535 increases locomotor activity in animal models of Parkinson׳s disease.

Physicochemical Properties

M.Wt 272.316
Formula C12H16N8
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

2-butyl-9-methyl-8-(2H-1,2,3-triazol-2-yl)-9H-purin-6-amine

References

1. Minetti P, et al. J Med Chem. 2005 Nov 3;48(22):6887-96.

2. Rose S, et al. Eur J Pharmacol. 2006 Sep 28;546(1-3):82-7.

3. Rose S, et al. Brain Res. 2007 Feb 16;1133(1):110-4.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: