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SUCNR1 inhibitor 20

Chemical Structure : SUCNR1 inhibitor 20

CAS No.: 2711753-52-3

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SUCNR1 inhibitor 20 (GPR91 antagonist)

Catalog No.: PC-72380Not For Human Use, Lab Use Only.

SUCNR1 inhibitor 20 is a potent, selective inhibitor (antagonist) of GPCR SUCNR1 (succinate receptor 1/GPR91) with IC50 of 88 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    SUCNR1 inhibitor 20 is a potent, selective inhibitor (antagonist) of GPCR SUCNR1 (succinate receptor 1/GPR91) with IC50 of 88 nM.
    SUCNR1 (GPR91) senses the citric cycle intermediate succinate and is implicated in various pathological conditions such as rheumatoid arthritis, liver fibrosis, or obesity.

    Physicochemical Properties

    M.Wt 518.917
    Formula C26H22ClF3N2O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (R)-2-(2-(4'-chloro-2,2'-difluoro-5'-(piperidin-3-yloxy)-[1,1'-biphenyl]-3-carboxamido)-5-fluorophenyl)acetic acid

    References

    1. Juraj Velcicky, et al. J Med Chem. 2020 Sep 10;63(17):9856-9875.

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