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Chemical Structure : T-10418
Catalog No.: PC-22564Not For Human Use, Lab Use Only.
T-10418 is a potent, selective agonist of G protein-coupled receptor G2A (GPR132) with EC50 of 0.82 uM.
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T-10418 is a potent, selective agonist of G protein-coupled receptor G2A (GPR132) with EC50 of 0.82 uM.
T-10418 exhibits higher potency than the reference and natural ligand 9-HODE and high selectivity among G protein-coupled receptors.
T-10418 has favorable activity, a clean selectivity profile, excellent solubility, and high metabolic stability, is a pharmacological tool to investigate the effects of G2A activation.
| M.Wt | 376.41 | |
| Formula | C22H20N2O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Hernandez-Olmos V, et al. J Med Chem. 2024 Jun 25. doi: 10.1021/acs.jmedchem.3c02164.
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