T-10418 | GPR132 agonist | Probechem Biochemicals

Chemical Structure : T-10418

T-10418 (T10418)

Catalog No.: PC-22564Not For Human Use, Lab Use Only.

T-10418 is a potent, selective agonist of G protein-coupled receptor G2A (GPR132) with EC50 of 0.82 uM.

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Biological Activity

T-10418 is a potent, selective agonist of G protein-coupled receptor G2A (GPR132) with EC50 of 0.82 uM.
T-10418 exhibits higher potency than the reference and natural ligand 9-HODE and high selectivity among G protein-coupled receptors.
T-10418 has favorable activity, a clean selectivity profile, excellent solubility, and high metabolic stability, is a pharmacological tool to investigate the effects of G2A activation.

Physicochemical Properties

M.Wt	376.41
Formula	C22H20N2O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(3-(pyridin-3-ylmethoxy)benzoyl)-D-phenylalanine

References

1. Hernandez-Olmos V, et al. J Med Chem. 2024 Jun 25. doi: 10.1021/acs.jmedchem.3c02164.

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T-10418 (T10418)

Biological Activity

Physicochemical Properties

References

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