TAK-901 |CAS:934541-31-8 Probechem Biochemicals

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Chemical Structure : TAK-901

CAS No.: 934541-31-8

TAK-901 (TAK901;TAK 901)

Catalog No.: PC-42912Not For Human Use, Lab Use Only.

TAK-901 is a multikinase inhibitor with IC50 of 21 nM and 15 nM for Aurora A/TPX2 and Aurora B/INCENP respectively.

Packing	Price	Stock
5 mg	$78	In stock
10 mg	$118	In stock
25 mg	$198	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

TAK-901 is a multikinase inhibitor with IC50 of 21 nM and 15 nM for Aurora A/TPX2 and Aurora B/INCENP respectively.
TAK-901 inhibits 56 kinases(IC50< 100 nM).
TAK-901 inhibits kinds of cancer cell lines with EC50s of 40-500 nM.
TAK-901 suppresses cellular histone H3 phosphorylation and induced polyploidy.

Physicochemical Properties

M.Wt	504.6437
Formula	C28H32N4O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	9H-Pyrido[2,3-b]indole-7-carboxamide, 5-[3-(ethylsulfonyl)phenyl]-3,8-dimethyl-N-(1-methyl-4-piperidinyl)-

References

1. Farrell P, et al. Mol Cancer Ther. 2013 Apr;12(4):460-70.

2. Murai S, et al. Anticancer Res. 2017 Feb;37(2):437-444.

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TAK-901 (TAK901;TAK 901)

Biological Activity

Physicochemical Properties

References

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