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Chemical Structure : TAK-901
CAS No.: 934541-31-8
Catalog No.: PC-42912Not For Human Use, Lab Use Only.
TAK-901 is a multikinase inhibitor with IC50 of 21 nM and 15 nM for Aurora A/TPX2 and Aurora B/INCENP respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $78 | In stock | |
| 10 mg | $118 | In stock | |
| 25 mg | $198 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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TAK-901 is a multikinase inhibitor with IC50 of 21 nM and 15 nM for Aurora A/TPX2 and Aurora B/INCENP respectively.
TAK-901 inhibits 56 kinases(IC50< 100 nM).
TAK-901 inhibits kinds of cancer cell lines with EC50s of 40-500 nM.
TAK-901 suppresses cellular histone H3 phosphorylation and induced polyploidy.
| M.Wt | 504.6437 | |
| Formula | C28H32N4O3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
9H-Pyrido[2,3-b]indole-7-carboxamide, 5-[3-(ethylsulfonyl)phenyl]-3,8-dimethyl-N-(1-methyl-4-piperidinyl)- |
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1. Farrell P, et al. Mol Cancer Ther. 2013 Apr;12(4):460-70.
2. Murai S, et al. Anticancer Res. 2017 Feb;37(2):437-444.
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