Chemical Structure : TCS-OX2-29
CAS No.:
372523-75-6
TCS-OX2-29
(TCS OX2 29)
Catalog No. : PC-42159Not For Human Use, Lab Use Only.
TCS-OX2-29 is a potent, selective orexin-2 receptor (OX2R) antagonist with IC50 of 40 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4215901
Biological Activity
TCS-OX2-29 is a potent, selective orexin-2 receptor (OX2R ) antagonist with IC50 of 40 nM.
Physicochemical Properties
M.Wt
397.5105
Formula
C23H31N3O3
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
1-Butanone, 1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-, (2S)-
References
1. Hirose M, et al. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4497-9.
2. Urbańska A, et al. J Mol Neurosci. 2012 Jan;46(1):10-7.
3. Huang SC, et al. J Pharmacol Exp Ther. 2010 Aug;334(2):522-9.
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