Chemical Structure : TM-04-176-01
CAS No.: 2428737-31-7
Catalog No.: PC-38271Not For Human Use, Lab Use Only.
TM-04-176-01 (PI5P4K inhibitor 13) is a selective pan-PI5P4K covalent inhibitor with IC50 of 2.0/13 uM against PI5P4Kα/β, 100% inhibition of PI5P4Kγ at 1 uM (Kd=3.4 nM).
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|---|---|---|---|
| 5 mg | $218 | In stock | |
| 10 mg | $348 | In stock | |
| 25 mg | $548 | In stock | |
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TM-04-176-01 (PI5P4K inhibitor 13) is a selective pan-PI5P4K covalent inhibitor with IC50 of 2.0/13 uM against PI5P4Kα/β, 100% inhibition of PI5P4Kγ at 1 uM (Kd=3.4 nM).
| M.Wt | 363.435 | |
| Formula | C20H17N3O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
N-(4-(5-(1H-indol-4-yl)pyridin-3-yl)phenyl)methanesulfonamide |
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1. Helen K Boffey, et al. J Med Chem. 2022 Feb 11. doi: 10.1021/acs.jmedchem.1c01819.

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