TM38837 | CB1 inverse agonist | Probechem Biochemicals

Chemical Structure : TM38837

Catalog No.: PC-22545Not For Human Use, Lab Use Only.

TM38837 is a potent, selective peripheral cannabinoid receptor 1 (CB1) inverse agonist with IC50 of 24 nM, 200-fold selective over CB2 receptor.

Packing	Price	Stock	Quantity
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

Get Quotation Now

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

TM38837 is a potent, selective peripheral cannabinoid receptor 1 (CB1) inverse agonist with IC50 of 24 nM, 200-fold selective over CB2 receptor.

M.Wt	586.40
Formula	C27H20Cl2F3N7O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(2-Chlorophenyl)-5-(4-chlorophenyl)-4-(2H-tetrazol-5-ylmethyl)-N-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]-1H-pyrazole-3-carboxamide

1. Micale V, et al. Front Pharmacol. 2019 Mar 20;10:207.

2. Högberg T, et al. Bioorg Med Chem Lett. 2024 Jan 15;98:129572.