TP-238 | 2415263-04-4 Probechem Biochemicals

Chemical Structure : TP-238

TP-238 (TP238)

Catalog No.: PC-35848Not For Human Use, Lab Use Only.

TP-238 (TP238) is a CECR2/BPTF bromodomains chemical probe with IC50 of 30 nM against CECR2 and 350 nM against BPTF in an alphascreen assay, KD of 10 nM for CECR2 and 120nM for BPTF in ITC assays.

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Biological Activity

TP-238 (TP238) is a CECR2/BPTF bromodomains chemical probe with IC50 of 30nM against CECR2 and 350 nM against BPTF in an alphascreen assay, KD of 10 nM for CECR2 and 120 nM for BPTF in ITC assays.
TP-238 has been profiled against the panel of 338 kinases and showed no activity at 1 uM, the closest off-target bromodomain inhibition is BRD9 with IC50 of 1.4 uM.

Physicochemical Properties

M.Wt	458.581
Formula	C22H30N6O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(3-(1H-pyrazol-1-yl)propyl)-6-(4-(3-(dimethylamino)propoxy)phenyl)-2-(methylsulfonyl)pyrimidin-4-amine

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TP-238 (TP238)

Biological Activity

Physicochemical Properties

References

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