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Chemical Structure : TRPM5 agonist 64
Catalog No.: PC-22256Not For Human Use, Lab Use Only.
TRPM5 agonist 64 is a potent, selective TRPM5 agonist with pEC50 of 7.8 and .1 for mTRPM5 and hTRPM5, respectively.
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TRPM5 agonist 64 is a potent, selective TRPM5 agonist with pEC50 of 7.8 and .1 for mTRPM5 and hTRPM5, respectively.
TRPM5 agonist 64 shows high selectivity (>100-fold) over hTRPM8/hTRPV1/hTRPV4/hTRPA1/hTRPM4 (pEC50, <4.8/<4.8/<4.8/5.5/5.5).
TRPM5 agonist 64 shows a statistically significant increase of the fecal parameters after oral administration at 100 mg/kg.
| M.Wt | 316.22 | |
| Formula | C11H7Cl2N3S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Alessio Barilli, et al. J Med Chem. 2021 May 13;64(9):5931-5955.
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