TRPV6 inhibitor cis-22a

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Chemical Structure : TRPV6 inhibitor cis-22a

Catalog No.: PC-25398Not For Human Use, Lab Use Only.

TRPV6 inhibitor cis-22a is a potent, selective inhibitor of TRPV6 calcium channel with IC50 of 0.32 uM, shows high selectivity against other calcium channels and related TRP targets, selectively reduces cancer cell growth on TRPV6 positive (T47D) breast cancer cells.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Physicochemical Properties

M.Wt	335.50
Formula	C22H29N3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-[cis-4-(3-Methylphenyl)cyclohexyl]-4-(3-pyridinyl)piperazine

References

1. Simonin C, et al. Angew. Chem. Int. Ed. Engl. 54, 14748–14752 (2015).

2. Bhardwaj R, et al. Sci Adv. 2020 Nov 27;6(48):eabe1508.

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