TUG-1958 | GPR43 antagonist | Probechem Biochemicals

Chemical Structure : TUG-1958

TUG-1958 (TUG1958)

Catalog No.: PC-24798Not For Human Use, Lab Use Only.

TUG-1958 is a potent, selective antagonist of GPR43 (FFA2R, free fatty acid receptor 2) with pIC50 of 7.41 uM (hFFA2) in [35S]GTPγS-based binding assays.

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Biological Activity

TUG-1958 is a potent, selective antagonist of GPR43 (FFA2R, free fatty acid receptor 2) with pIC50 of 7.41 uM (hFFA2) in [35S]GTPγS-based binding assays.
TUG-1958 is completely selective over the related receptor FFA3 with no sign of activity up to 100 μM.
TUG-1958 has excellent solubility and favorable pharmacokinetic properties.

Physicochemical Properties

M.Wt	397.37
Formula	C20H19F4NO3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-4-(2-(3-fluorophenyl)acetamido)-5-(4-(trifluoromethyl)phenyl)pentanoic acid

References

1. Højgaard Hansen A, et al. ChemMedChem. 2021 Nov 5;16(21):3326-3341.

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TUG-1958 (TUG1958)

Biological Activity

Physicochemical Properties

References

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