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Trotabresib

Chemical Structure : Trotabresib

CAS No.: 1706738-98-8

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Trotabresib (CC-90010, CC90010, QC5487)

Catalog No.: PC-38040Not For Human Use, Lab Use Only.

Trotabresib (CC90010) is a reversible and orally active BET bromodomain inhibitor, shows significant antiproliferative activity in glioblastoma cells and patient-derived xenograft models as monotherapy and in combination with temozolomide (TMZ).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Trotabresib (CC90010) is a reversible and orally active BET bromodomain inhibitor, shows significant antiproliferative activity in glioblastoma cells and patient-derived xenograft models as monotherapy and in combination with temozolomide (TMZ).

Physicochemical Properties

M.Wt 383.462
Formula C21H21NO4S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1(2H)-Isoquinolinone, 4-(2-(cyclopropylmethoxy)-5-(methylsulfonyl)phenyl)-2-methyl-

References

1. Moreno V, et al. Ann Oncol. 2020 Jun;31(6):780-788.

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