Chemical Structure : Tulmimetostat
CAS No.: 2567686-02-4
Catalog No.: PC-73451Not For Human Use, Lab Use Only.
Tulmimetostat (CPI-0209) is a potent, selective, orally available EZH2 inhibitor with Ki of 140 fM by kinetic analyses and Ki 180 fM by thermal shift assays.
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10 mg | $458 | In stock | |
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M.Wt | 562.122 | |
Formula | C28H36ClN3O5S | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
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Chemical Name/SMILES |
(2R)-7-cloro-2,4-dimetil-N-{[6-metil-4-(metilsulfanil)-2- oxo-1,2-dihidropiridin-3-il]metil}-2-[trans-4-(3- metoxiazetidin-1-il)ciclohexil]-2H-1,3-benzodioxol-5- carboxamida |
1. Patent WO2021016409 A1.
2. Keller PJ, et al. Cancer Res. 2024 Jun 4. doi: 10.1158/0008-5472.CAN-24-0398.
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