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UNC0224

Chemical Structure : UNC0224

CAS No.: 1197196-48-7

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UNC0224 (UNC 0224, UNC-0224)

Catalog No.: PC-42740Not For Human Use, Lab Use Only.

UNC0224 (UNC-0224) is a potent, selective G9a/GLP inhibitor with IC50 of 57 nM and 58 nM in biochemical assays.

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5 mg $78 In stock
10 mg $118 In stock
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50 mg $358 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

UNC0224 (UNC-0224) is a potent, selective G9a/GLP inhibitor with IC50 of 57 nM and 58 nM in biochemical assays.
UNC0224 dispalys >1000-fold selectivity for G9a over SET7/9, SET8, PRMT3 and JMJD2E (IC50>4 uM).

Physicochemical Properties

M.Wt 485.6653
Formula C26H43N7O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-Quinazolinamine, 7-[3-(dimethylamino)propoxy]-2-(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6-methoxy-N-(1-methyl-4-piperidinyl)-

References

1. Liu F, et al. J Med Chem. 2010 Aug 12;53(15):5844-57.

2. Liu F, et al. J Med Chem. 2009 Dec 24;52(24):7950-3.

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