Chemical Structure : UNC0224
CAS No.: 1197196-48-7
Catalog No.: PC-42740Not For Human Use, Lab Use Only.
UNC0224 (UNC-0224) is a potent, selective G9a/GLP inhibitor with IC50 of 57 nM and 58 nM in biochemical assays.
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UNC0224 (UNC-0224) is a potent, selective G9a/GLP inhibitor with IC50 of 57 nM and 58 nM in biochemical assays.
UNC0224 dispalys >1000-fold selectivity for G9a over SET7/9, SET8, PRMT3 and JMJD2E (IC50>4 uM).
M.Wt | 485.6653 | |
Formula | C26H43N7O2 | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
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Chemical Name/SMILES |
4-Quinazolinamine, 7-[3-(dimethylamino)propoxy]-2-(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6-methoxy-N-(1-methyl-4-piperidinyl)- |
1. Liu F, et al. J Med Chem. 2010 Aug 12;53(15):5844-57.
2. Liu F, et al. J Med Chem. 2009 Dec 24;52(24):7950-3.
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