Chemical Structure : UNC0379
CAS No.:
1620401-82-2
UNC0379
(UNC 0379, UNC-0379)
Catalog No. : PC-42983Not For Human Use, Lab Use Only.
UNC0379 is a selective, substrate-competitive inhibitor of lysine methyltransferase SETD8 with IC50 of 7.3 uM.
Packing Price Stock Quantity 10 mg $88 In stock 0 1 2 3 4 5 25 mg $138 In stock 0 1 2 3 4 5 50 mg $218 In stock 0 1 2 3 4 5 100 mg $358 In stock 0 1 2 3 4 5 250 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4298301
Biological Activity
UNC0379 is a selective, substrate-competitive inhibitor of lysine methyltransferase SETD8 with IC50 of 7.3 uM.
Physicochemical Properties
M.Wt
413.5563
Formula
C23H35N5O2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
4-Quinazolinamine, 6,7-dimethoxy-2-(1-pyrrolidinyl)-N-[5-(1-pyrrolidinyl)pentyl]-
References
1. Ma A, et al. J Med Chem.
2. Ma A, et al. Medchemcomm.
3. Veschi V, et al. Cancer Cell.
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