USP7-866 | USP7 inhibitor | Probechem Biochemicals

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Chemical Structure : USP7-866

USP7-866 (USP 7-866)

Catalog No.: PC-38192Not For Human Use, Lab Use Only.

USP7-866 is a novel potent selective inhibitor of USP7 with IC50 of 0.18 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

USP7-866 is a novel potent selective inhibitor of USP7 with IC50 of 0.18 nM.
USP7-866 inhibited the growth of p53-mutant small cell lung cancer cell line H526 at a CC50 of 42 nM.

Physicochemical Properties

M.Wt	524.076
Formula	C28H30ClN3O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-((7-(5-chloro-3-methyl-2-(((3S,4R)-3-methylpiperidin-4-yl)oxy)phenyl)thieno[3,2-b]pyridin-2-yl)methyl)-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2,4-dione

References

1. Yamini M Ohol, et al. Mol Cancer Ther. 2020 Oct;19(10):1970-1980.

2. Paul R Leger, et al. J Med Chem. 2020 May 28;63(10):5398-5420.

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USP7-866 (USP 7-866)

Biological Activity

Physicochemical Properties

References

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