VU6001966 | mGlu2 NAM | Probechem Biochemicals

Chemical Structure : VU6001966

CAS No.: 2009052-76-8

VU6001966 (VU-6001966)

Catalog No.: PC-60939Not For Human Use, Lab Use Only.

VU 6001966 is a potent and selective, CNS penetrant mGlu2 negative allosteric modulator with IC50 of 78 nM.

Packing	Price	Stock
5 mg	$328	In stock
10 mg	$528	In stock
50 mg		Get quote
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

VU 6001966 is a potent and selective, CNS penetrant mGlu2 negative allosteric modulator with IC50 of 78 nM.
VU 6001966 shows no inhibition for mGlu3 (IC50>30 uM).
VU 6001966 represents an exciting lead series for potential mGlu2 PET tracer development.

Physicochemical Properties

M.Wt	326.331
Formula	C17H15FN4O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(4-fluorophenyl)-5-((1-methyl-1H-pyrazol-3-yl)methoxy)picolinamide

References

1. Bollinger KA, et al. ACS Med Chem Lett. 2017 Aug 3;8(9):919-924.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

VU6001966 (VU-6001966)

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.