VU6001966 | mGlu2 NAM | Probechem Biochemicals

Chemical Structure : VU6001966

VU6001966 (VU-6001966)

Catalog No.: PC-60939Not For Human Use, Lab Use Only.

VU 6001966 is a potent and selective, CNS penetrant mGlu2 negative allosteric modulator with IC50 of 78 nM.

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Biological Activity

VU 6001966 is a potent and selective, CNS penetrant mGlu2 negative allosteric modulator with IC50 of 78 nM.
VU 6001966 shows no inhibition for mGlu3 (IC50>30 uM).
VU 6001966 represents an exciting lead series for potential mGlu2 PET tracer development.

Physicochemical Properties

M.Wt	326.331
Formula	C17H15FN4O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(4-fluorophenyl)-5-((1-methyl-1H-pyrazol-3-yl)methoxy)picolinamide

References

1. Bollinger KA, et al. ACS Med Chem Lett. 2017 Aug 3;8(9):919-924.

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VU6001966 (VU-6001966)

Biological Activity

Physicochemical Properties

References

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