Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-GPCR-mGluR-VU6020933
VU6020933

Chemical Structure : VU6020933

CAS No.: 2839123-04-3

VU6020933 (VU 6020933)

Catalog No.: PC-22901Not For Human Use, Lab Use Only.

VU6020933 is a potent, selective, dual mGlu2/mGlu3 positive allosteric modulator with EC50 of 164/476 nM, respectively, potentiates group II mGlu receptor agonist Ca2+ signaling in PFC pyramidal cells.

Packing Price Stock Quantity
50 mg Get quote
100 mg Get quote
250mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

VU6020933 is a potent, selective, dual mGlu2/mGlu3 positive allosteric modulator with EC50 of 164/476 nM, respectively, potentiates group II mGlu receptor agonist Ca2+ signaling in PFC pyramidal cells.

Physicochemical Properties

M.Wt 445.53
Formula C25H32FNO5
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

5-(4-(4-(3,3-dimethylbutanoyl)-3-hydroxy-2-methylphenoxy)butoxy)-2-fluoro-N-methylbenzamide

References

1. Yousuke Yamada, et al. Bioorg Med Chem Lett. 2021 Oct 15:50:128342.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: