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VUF15485

Chemical Structure : VUF15485

CAS No.: 2800877-68-1

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VUF15485 (VUF-15485, VUF 15485)

Catalog No.: PC-21785Not For Human Use, Lab Use Only.

VUF15485 is a small-molecule agonist of the atypical chemokine receptor ACKR3 (CXCR7) with binding pIC50 of 8.3, and pEC50 of 7.6 in BRET-based β-arrestin2 recruitment assay.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    VUF15485 is a small-molecule agonist of the atypical chemokine receptor ACKR3 (CXCR7) with binding pIC50 of 8.3, and pEC50 of 7.6 in BRET-based β-arrestin2 recruitment assay.
    VUF15485 is highly selective for ACKR3 against a chemokine receptor panel (agonist and antagonist mode).

    Physicochemical Properties

    M.Wt 470.59
    Formula C27H35FN2O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (R,E)-N-(3-(2-fluorophenyl)-2-methylallyl)-3,4,5-trimethoxy-N-(2-(1-methylpyrrolidin-2-yl)ethyl)benzamide

    References

    1. Aurelien Zarca, et al. Mol Pharmacol. 2024 Feb 12:MOLPHARM-AR-2023-000835.

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