VUF15485 | ACKR3 agonist | Probechem Biochemicals

Chemical Structure : VUF15485

VUF15485 (VUF 15485)

Catalog No.: PC-21785Not For Human Use, Lab Use Only.

VUF15485 is a small-molecule agonist of the atypical chemokine receptor ACKR3 with binding pIC50 of 8.3, and pEC50 of 7.6 in BRET-based β-arrestin2 recruitment assay.

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Biological Activity

VUF15485 is a small-molecule agonist of the atypical chemokine receptor ACKR3 with binding pIC50 of 8.3, and pEC50 of 7.6 in BRET-based β-arrestin2 recruitment assay.
VUF15485 is highly selective for ACKR3 against a chemokine receptor panel (agonist and antagonist mode).

Physicochemical Properties

M.Wt	470.59
Formula	C27H35FN2O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R,E)-N-(3-(2-fluorophenyl)-2-methylallyl)-3,4,5-trimethoxy-N-(2-(1-methylpyrrolidin-2-yl)ethyl)benzamide

References

1. Aurelien Zarca, et al. Mol Pharmacol. 2024 Feb 12:MOLPHARM-AR-2023-000835.

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VUF15485 (VUF 15485)

Biological Activity

Physicochemical Properties

References

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