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WDR5-0103

Chemical Structure : WDR5-0103

CAS No.: 890190-22-4

WDR5-0103 (WD-Repeat Protein 5-0103)

Catalog No.: PC-45617Not For Human Use, Lab Use Only.

A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.

Packing Price Stock Quantity
5 mg (Free Sample) $28 In stock
10 mg $78 In stock
25 mg $138 In stock
50 mg $218 In stock
100 mg Get quote

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

WDR5-0103 is a potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.
WDR5-0103 inhibits the catalytic activity of MLL1 complex with IC50 value of 5.4 uM.

Physicochemical Properties

M.Wt 383.4409
Formula C21H25N3O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 40 mg/mL

Chemical Name/SMILES

Benzoic acid, 3-[(3-methoxybenzoyl)amino]-4-(4-methyl-1-piperazinyl)-, methyl ester

References

1. Li DD, et al. Bioorg Med Chem. 2016 Nov 15;24(22):6109-6118.

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