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WDR5 WBM site inhibitor 7k

Chemical Structure : WDR5 WBM site inhibitor 7k

CAS No.: 2581117-13-5

WDR5 WBM site inhibitor 7k

Catalog No.: PC-21832Not For Human Use, Lab Use Only.

WDR5 WBM site inhibitor 7k is a selective small molecule inhibitor of WDR5 WBM binding site with Ki of 107 nM, inhibits lncRNA-WDR5 complex formation.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

WDR5 WBM site inhibitor 7k is a selective small molecule inhibitor of WDR5 WBM binding site with Ki of 107 nM, inhibits lncRNA-WDR5 complex formation.
WDR5 WBM site inhibitor 7k shows no activity against WDR5 WIN site binding.
WDR5 WBM site inhibitor 7k reduces cMYC enrichment in WDR5 pull-down experiments, downregulates HOTTIP.

Physicochemical Properties

M.Wt 514.78
Formula C19H17BrClN3O5S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

3-((5-bromo-3-chloro-2-hydroxyphenyl)sulfonamido)-5-(1-cyanocyclobutyl)-2-hydroxy-N-methylbenzamide

References

1. Chang JY, et al. RSC Med Chem. 2024 Jan 10;15(2):636-640.

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