WHI-P131 | JAK3 inhibitor | Probechem Biochemicals

Chemical Structure : WHI-P131

CAS No.: 202475-60-3

Catalog No.: PC-21425Not For Human Use, Lab Use Only.

WHI-P131 (JANEX-1) is a potent and selective JAK3 inhibitor with Ki of 2.3 uM and IC50 of 78 uM, with no activity agianst JAK1 and JAK2.

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Biological Activity

WHI-P131 (JANEX-1) is a potent and selective JAK3 inhibitor with Ki of 2.3 uM and IC50 of 78 uM, with no activity agianst JAK1 and JAK2.

M.Wt	297.31
Formula	C16H15N3O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-((6,7-Dimethoxyquinazolin-4-yl)amino)phenol

1. Uckun FM, et al. Clin Cancer Res. 1999 Oct;5(10):2954-62.

2. Malaviya R, et al. J Biol Chem. 1999 Sep 17;274(38):27028-38.

3. Narla RK, et al. Clin Cancer Res. 1998 Oct;4(10):2463-71.