WHI-P97 | JAK3 inhibitor | Probechem Biochemicals

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Chemical Structure : WHI-P97

CAS No.: 211555-05-4

WHI-P97 (WHI-P-97;WHI P97)

Catalog No.: PC-42802Not For Human Use, Lab Use Only.

WHI-P97 is a potent, specific JAK3 inhibitor with Ki of 0.6-2.3 uM.

Packing	Price	Stock
10 mg	$128	In stock
25 mg	$218	In stock
50 mg	$368	In stock
100 mg		Get quote

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

WHI-P97 is a potent, specific JAK3 inhibitor with Ki of 0.6-2.3 uM.
WHI-P97 inhibits the translocation of 5-lipoxygenase (5-LO) from the nucleoplasm to the nuclear membrane and inhibits mast cell leukotriene synthesis in vitro.
WHI-P97 shows promising biological activity in mouse model of allergic asthma.

Physicochemical Properties

M.Wt	455.1007
Formula	C16H13Br2N3O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Phenol, 2,6-dibromo-4-[(6,7-dimethoxy-4-quinazolinyl)amino]-

References

1. Malaviya R, et al. J Pharmacol Exp Ther. 2000 Dec;295(3):912-26.

2. Sudbeck EA, et al. Clin Cancer Res. 1999 Jun;5(6):1569-82.

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WHI-P97 (WHI-P-97;WHI P97)

Biological Activity

Physicochemical Properties

References

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