Y08284 | CBP/p300 inhibitor | Probechem Biochemicals

Chemical Structure : Y08284

Catalog No.: PC-22485Not For Human Use, Lab Use Only.

Y08284 is a potent, selective CBP/p300 bromodomain inhibitor with IC50 of 4.21 nM (CBP bromodomain) in HTRF assays.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Y08284 is a potent, selective CBP/p300 bromodomain inhibitor with IC50 of 4.21 nM (CBP bromodomain) in HTRF assays.

M.Wt	476.51
Formula	C26H25FN4O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-Acetyl-N-(3-(1-cyclopropyl-1H-pyrazol-4-yl)-2-fluoro-5-(1-hydroxyethyl)phenyl)-7-methoxyindolizine-1-carboxamide

1. Qiuping Xiang, et al. J Med Chem. 2022 Jan 13;65(1):785-810.