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Chemical Structure : ZINC621433144
Catalog No.: PC-20978Not For Human Use, Lab Use Only.
ZINC621433144 is a Gi-biased, high-affinity full agonist of dopamine D4 receptor with Ki of 4.3 nM and cAMP EC50 of 0.18 nM.
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ZINC621433144 is a Gi-biased, high-affinity full agonist of dopamine D4 receptor with Ki of 4.3 nM and cAMP EC50 of 0.18 nM.
ZINC621433144 displays no affinity for D2 and D3 receptors.
ZINC621433144 shows EC50 of 0.56 and 2.3 nM in Gi BRET and Arrestin BRET assays, respectively.
| M.Wt | 301.43 | |
| Formula | C18H27N3O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Jiankun Lyu, et al. Nature. 2019 Feb;566(7743):224-229.
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