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ZK-216348

Chemical Structure : ZK-216348

CAS No.: 669073-68-1

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ZK-216348 (ZK216348)

Catalog No.: PC-35001Not For Human Use, Lab Use Only.

ZK-216348 is a potent, selective, dissociated glucocorticoid receptor agonist with pIC50 of 7.7, shows selectivity over other nuclear hormone receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    ZK-216348 is a potent, selective, dissociated glucocorticoid receptor agonist with pIC50 of 7.7, shows selectivity over other nuclear hormone receptors.

    Physicochemical Properties

    M.Wt 476.45
    Formula C24H23F3N2O5
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    4-(2,3-dihydro-1-benzofuran-7-yl)-2-hydroxy-4-methyl-N-(4-methyl-1-oxo-2,3-benzoxazin-6-yl)-2-(trifluoromethyl)pentanamide

    References

    1. Schäcke H, et al. Proc Natl Acad Sci U S A. 2004 Jan 6;101(1):227-32.

    2. Jaroch S, et al. Bioorg Med Chem Lett. 2010 Oct 1;20(19):5835-8.

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