mTOR-IN-1 |CAS:1207358-59-5 Probechem Biochemicals

Chemical Structure : mTOR-IN-1

CAS No.: 1207358-59-5

mTOR-IN-1

Catalog No.: PC-45461Not For Human Use, Lab Use Only.

mTOR-IN-1 is a potent and selective mTOR inhibitor with Ki of 1.5 nM.

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5 mg	$148	In stock
10 mg	$228	In stock
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Biological Activity

mTOR-IN-1 is a potent and selective mTOR inhibitor with Ki of 1.5 nM.
mTOR-IN-1 shows >500-fold selectivity over closely related PI3 kinases.
mTOR-IN-1 exhibits suitable mouse PK and demenstrates active in an NCI-PC3prostate cancer model; orally bioavailable.

Physicochemical Properties

M.Wt	474.5581
Formula	C25H30N8O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Urea, N-ethyl-N'-[4-[5,6,7,8-tetrahydro-4-[(3S)-3-methyl-4-morpholinyl]-7-(2-pyrimidinyl)pyrido[3,4-d]pyrimidin-2-yl]phenyl]-

References

1. Koehler MF, et al. J Med Chem. 2012 Dec 27;55(24):10958-71.

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mTOR-IN-1

Biological Activity

Physicochemical Properties

References

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