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Chemical Structure : DRAK2-IN-16
CAS No.: 871837-60-4
Catalog No.: PC-62719Not For Human Use, Lab Use Only.
DRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM, shows weak inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM)..
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $228 | In stock | |
| 10 mg | $378 | In stock | |
| 25 mg | $588 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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DRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM, shows weak inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM).
| M.Wt | 376.416 | |
| Formula | C21H20N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
N-((2Z,3E)-3-(hydroxyimino)-2'-oxo-[2,3'-biindolinylidene]-5'-yl)pentanamide |
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1. Jung ME, et al. Bioorg Med Chem Lett. 2016 Jun 1;26(11):2719-23.
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