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GR-64349

Chemical Structure : GR-64349

CAS No.: 137593-52-3

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GR-64349 (GR64349)

Catalog No.: PC-63098Not For Human Use, Lab Use Only.

GR-64349 is a potent and selective tachykinin NK2 receptor (NK2R) agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GR-64349 is a potent and selective tachykinin NK2 receptor (NK2R) agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.

Physicochemical Properties

M.Wt 921.12
Formula C42H68N10O11S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

KDSFVGLM (Modifications: Leu-7 = R-γ-lactam-Leu, Met-8 = C-terminal amide)

References

1. Deal MJ, et al. J Med Chem. 1992 Oct 30;35(22):4195-204.

2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.

3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.

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