GSK-575594A |CAS:909418-68-4 Probechem Biochemicals

Chemical Structure : GSK-575594A

GSK-575594A (GSK575594A)

Catalog No.: PC-63115Not For Human Use, Lab Use Only.

GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0).

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Biological Activity

GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0).
GSK-575594A activates human GPR55 but not rodent GPR55, and is inactive at cannabinoid receptors.

Physicochemical Properties

M.Wt	471.523
Formula	C24H23F2N3O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	[4-(4-amino-2-fluorophenyl)piperazin-1-yl]-[2-(4-fluorophenyl)-5-methylsulfonylphenyl]methanone

References

1. Brown AJ, et al. J Pharmacol Exp Ther. 2011 Apr;337(1):236-46.

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GSK-575594A (GSK575594A)

Biological Activity

Physicochemical Properties

References

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