Chemical Structure : GSK-575594A
Catalog No.: PC-63115Not For Human Use, Lab Use Only.
GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0).
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GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0).
GSK-575594A activates human GPR55 but not rodent GPR55, and is inactive at cannabinoid receptors.
M.Wt | 471.523 | |
Formula | C24H23F2N3O3S | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Brown AJ, et al. J Pharmacol Exp Ther. 2011 Apr;337(1):236-46.
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