You are here:Home-Chemical Inhibitors & Agonists-GPCR-GPR55-GSK-575594A
GSK-575594A

Chemical Structure : GSK-575594A

CAS No.: 909418-68-4

GSK-575594A (GSK575594A)

Catalog No.: PC-63115Not For Human Use, Lab Use Only.

GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0).

Packing Price Stock Quantity
50 mg Get quote
100 mg Get quote
200 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    GSK-575594A is a potent, selective GPR55 agonist with pEC50 of 6.8 at GPR55 in yeast assay, displays 60-fold selective for GPR55 over GlyT1 (pIC50=5.0).
    GSK-575594A activates human GPR55 but not rodent GPR55, and is inactive at cannabinoid receptors.

    Physicochemical Properties

    M.Wt 471.523
    Formula C24H23F2N3O3S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    [4-(4-amino-2-fluorophenyl)piperazin-1-yl]-[2-(4-fluorophenyl)-5-methylsulfonylphenyl]methanone

    References

    1. Brown AJ, et al. J Pharmacol Exp Ther. 2011 Apr;337(1):236-46.

    Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    Contact Us sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    Get Quote

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • Additional Information: