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Chemical Structure : TSU-68
CAS No.: 252916-29-3
Catalog No.: PC-42630Not For Human Use, Lab Use Only.
TSU-68 (Orantinib, SU6668) is a small-molecule, ATP-competitive inhibitor of angiogenic related RTKs KDR, PDGFRβ, FGFR1.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $88 | In stock | |
| 25 mg | $128 | In stock | |
| 50 mg | $198 | In stock | |
| 100 mg | Get quote |
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TSU-68 (Orantinib, SU6668) is a small-molecule, ATP-competitive inhibitor of angiogenic related RTKs KDR, PDGFRβ, FGFR1.
TSU-68 inhibits receptor tyrosine phosphorylation and mitogenesis after stimulation of cells by appropriate ligands.
TSU-68 significant growth inhibition of a diverse panel of human tumor xenografts after oral or i.p. administration.
| M.Wt | 310.3471 | |
| Formula | C18H18N2O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 28 mg/mL |
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| Chemical Name/SMILES |
1H-Pyrrole-3-propanoic acid, 5-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-2,4-dimethyl- |
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1. Laird AD, et al. Cancer Res. 2000 Aug 1;60(15):4152-60.
2. Shaheen RM, et al. Cancer Res. 2001 Feb 15;61(4):1464-8.
3. Marzola P, et al. Clin Cancer Res. 2004 Jan 15;10(2):739-50.
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