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VPC-23019

Chemical Structure : VPC-23019

CAS No.: 449173-19-7

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VPC-23019 (VPC23019)

Catalog No.: PC-70075Not For Human Use, Lab Use Only.

VPC-23019 is a competitive S1P receptor antagonist with pKi of 7.86 and 5.93 for S1P1 and S1P3, respectively, in radioligand binding assays.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

VPC-23019 is a competitive S1P receptor antagonist with pKi of 7.86 and 5.93 for S1P1 and S1P3, respectively, in radioligand binding assays.
VPC-23019 increases the concentration-dependent vasoconstriction to S1P in both rat and mouse basilar arteries with intact endothelium.

Physicochemical Properties

M.Wt 372.4
Formula C17H29N2O5P
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(R)-2-amino-3-((3-octylphenyl)amino)-3-oxopropyl dihydrogen phosphate

References

1. Davis MD, et al. J Biol Chem. 2005 Mar 18;280(11):9833-41.

2. El-Shewy HM, et al. J Biol Chem. 2006 Oct 20;281(42):31399-407.

3. Salomone S, et al. Br J Pharmacol. 2008 Jan;153(1):140-7.

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