Cat. No. |
Product Name |
Information |
PC-42257 |
GMX1778
NAMPT inhibitor
|
GMX1778 (CHS-828) is a potent, specific, competitive NAMPT inhibitor with Kd of 120 nM, enzyme IC50 of <25 nM. |
PC-45883 |
FK-866
NAMPT inhibitor
|
FK-866 (Daporinad, APO-866) is a potent, highly specific nicotinamide phosphoribosyltransferase (NAMPT) inhibitor with Ki of 0.4 nM. |
PC-22010 |
LZFPN-90
NAMPT/PD-L1 inhibitor
|
LZFPN-90 (LZ90) is a potent, dual NAMPT/PD-L1 targeting inhibitor with IC50 of 13 nM/28 nM for PD-1/PD-L1 and NAMPT, respectively. |
PC-21428 |
A4276
NAMPT inhibitor
|
A4276 is a novel orally bioavailable NAMPT inhibitor with IC50 of 492 nM for inhibiting NAMPT enzymatic activity, shows high selectivity for NAPRT-deficient lung cancer cell lines. |
PC-21052 |
MM201
NAMPT inhibitor
|
MM201 is a novel potent nicotinamide phosphoribosyltransferase (NAMPT) inhibitor with IC50 of 74.3 nM in in vitro biochemical assays. |