| Cat. No. |
Product Name |
Information |
| PC-26906 |
CX1003
MET/VEGFR-2 inhibitor
|
CX1003 is a novel multitargeted receptor tyrosine kinase inhibitor targeting MET and VEGFR types 2 (VEGFR-2, KDR), also possesses inhibitory activities against several other kinases, such as Ret. |
| PC-24709 |
MET transcriptional inhibitor C3
CAS 3082125-66-1
|
MET transcriptional inhibitor C3 is a potent MET transcriptional inhibitor, efficiently binds to the G-quadruplex (G4, Kd=73.5 nM) in the MET promoter and suppresses the expression of c-Met. |
| PC-22805 |
MET inhibitor 13
MET inhibitor
|
MET inhibitor 13 is a potent, selective and mutant-active MET kinase inhibitor with IC50 of 6/6 nM for D1228N/exon Δ14 enzyme, and 90/15/5 nM for F1200I/L1995 V/Y1230H mutants respectively. |