Cat. No. |
Product Name |
Information |
PC-42835 |
SGX-523
|
SGX-523 is a potent, selective ATP-competitive inhibitor of MET receptor tyrosine kinase with IC50 of 4 nM, does not inhibit RON and a panel of kinases. |
PC-42833 |
PF-04217903 methanesulfonate
|
PF-04217903 is a potent, selective, ATP-competitive c-Met kinase inhibitor with Ki of 4.8 nM, inhibits HGF-stimulated tyrosine phosphorylation of wild type c-Met with IC50 of 7.3 nM in cell-based assays. |
PC-60929 |
MET inhibitor Compound 1
|
A novel potent, selective orally bioavailable MET tyrosine kinase inhibitor with IC50 of <1 nM and 12 nM for unphosphorylated and phosphorylaed MET, respectively. |
PC-60656 |
SOMG-833
|
A potent, selective, ATP-competitive c-MET inhibitor with IC50 of 0.93 nM. |
PC-60463 |
SAR 125844
|
A potent, highly selective, ATP-competitive MET receptor tyrosine kinase inhibitor with IC50 of 4.2 nM. |