ARN-3261 | Probechem Biochemicals

Chemical Structure : ARN-3261

ARN-3261 (ARN 3261;ARN3261)

Catalog No.: PC-61952Not For Human Use, Lab Use Only.

ARN-3261 is a potent, selective, orally available salt inducible kinase SIK2 and SIK3 inhibitor with IC50 of 11 nM and 19 nM, respectively.

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Biological Activity

ARN-3261 is a potent, selective, orally available salt inducible kinase SIK2 and SIK3 inhibitor with IC50 of 11 nM and 19 nM, respectively; specifically inhibits SIK2-expressed SKOv3 cells with IC50 of 92 nM; demonstrates effectivity against ovarian, breast cancer cell lines alone and in combination with Paclitaxel and Cisplatin; also inhibits ovarian tumor growth significantly in SKOv3 human ovarian cancer xenografts in mice.

Physicochemical Properties

M.Wt
Formula
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES

References

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ARN-3261 (ARN 3261;ARN3261)

Biological Activity

Physicochemical Properties

References

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