Cat. No. |
Product Name |
CAS No. |
Information |
PC-36096 |
Pizuglanstat
|
1244967-98-3 |
TAS-205 (Pizuglanstat, TAS205) is a potent, specific hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with IC50 of 55.8 nM, does not inhibit LPGDS at 100 uM. |
PC-36090 |
Crisdesalazine
|
927685-43-6 |
Crisdesalazine (AAD-2004, AAD2004) is a derivative of aspirin that inhibits microsomal PGE(2) synthase-1 (mPGES-1) activity in response to both LPS-treated BV2 cell with IC50 of 230 nM and recombinant human mPGES-1 protein with IC50 of 249 nM in vitro. |
PC-20005 |
mPGES-1 inhibitor UK-4b
|
2171000-87-4 |
mPGES-1 inhibitor UK-4b is a potent, hgihly selective and orally bioavailable inhibitor of human and mouse mPGES-1 enzymes with IC50 of 33 and 157 nM, respectively, effectively decreases carrageenan-stimulated PGE2 over-production. |
PC-49705 |
mPGES-1 inhibitor PBCH
|
2002435-92-7 |
PBCH is a selective small-molecule inhibitor of mPGES-1, which is potent and can effectively inhibit both human and rodent orthologs. |
PC-49642 |
TAS-204
|
920286-12-0 |
TAS-204 (TAS204) is a potent, specific hematopoietic prostaglandin D synthase (H-PGDS) inhibitor, inhibits recombinant human H-PGDS with IC50 of 24.0 nM. |
PC-49641 |
TAS-205 monohydrate
|
1584160-52-0 |
TAS-205 (Pizuglanstat, TAS205) is a potent, specific hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with IC50 of 55.8 nM, does not inhibit LPGDS at 100 uM. |
PC-49640 |
TFC-007
|
927878-49-7 |
TFC-007 (TFC007) is a potent, specific hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with IC50 of 83 nM. |