BRD4 degrader AT1 | BRD4 PROTAC | Probechem Biochemicals

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Chemical Structure : BRD4 degrader AT1

CAS No.: 2098836-45-2

BRD4 degrader AT1 (BRD4 PROTAC AT1)

Catalog No.: PC-35351Not For Human Use, Lab Use Only.

BRD4 degrader AT1 is a highly selective BRD4 degrader (PROTAC), exhibits highly selective depletion of BRD4 in cells with negligible activity against BRD2 and BRD3.

Packing	Price	Stock
1 mg	$118	In stock
5 mg	$288	In stock
10 mg	$488	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BRD4 degrader AT1 is a highly selective BRD4 degrader (PROTAC), exhibits highly selective depletion of BRD4 in cells with negligible activity against BRD2 and BRD3.

Physicochemical Properties

M.Wt	972.68
Formula	C48H58ClN9O5S3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S,4R)-1-((R)-2-acetamido-3-((6-(2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)hexyl)thio)-3-methylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide

References

1. Gadd MS, et al. Structural basis of PROTAC cooperative recognition for selective protein degradation. Nat Chem Biol. 2017 May;13(5):514-521.

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BRD4 degrader AT1 (BRD4 PROTAC AT1)

Biological Activity

Physicochemical Properties

References

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