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Chemical Structure : FAAH-IN-2
Catalog No.: PC-70218Not For Human Use, Lab Use Only.
A potent, selective, noncovalent FAAH inhibitor with IC50 of 28 nM toward human FAAH and 100 nM toward rat FAAH.
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A potent, selective, noncovalent FAAH inhibitor with IC50 of 28 nM toward human FAAH and 100 nM toward rat FAAH; demonstrates an excellent selectivity profile against a panel of cannabinoid related targets, including CB1, CB2, and VR1; demonstrates a unique nonmechanism-based inhibition of FAAH activity, which is distinct from almost all known FAAH inhibitors; shows excellent PK properties with a low clearance of 0.4 L/h/Kg and a high bioavailability of 92%.
| M.Wt | 421.266 | |
| Formula | C19H18BrFN2O3 | |
| Appearance | Solid | |
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| Solubility |
10 mM in DMSO |
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1. Min X, et al. Proc Natl Acad Sci U S A. 2011 May 3;108(18):7379-84.
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