NU-6300 |CAS: 2070015-09-5 Probechem Biochemicals

Chemical Structure : NU-6300

CAS No.: 2070015-09-5

NU-6300 (NU 6300;NU6300)

Catalog No.: PC-45559Not For Human Use, Lab Use Only.

NU-6300 is the first covalent, irreversible, ATP-Competitive CDK2 inhibitor with Ki of 6 nM.

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25 mg	$598	In stock
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Biological Activity

NU-6300 is the first covalent, irreversible, ATP-Competitive CDK2 inhibitor with Ki of 6 nM.
NU-6300 shows modest effect (GI50=8 uM) against human MCF-7 breast carcinoma cells.
NU-6300 inhibits Rb phosphorylation in Rb-positive SKUT-1B cells.

Physicochemical Properties

M.Wt	413.4933
Formula	C20H23N5O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	DMSO: ≥ 32 mg/mL
Chemical Name/SMILES	6-(cyclohexylmethoxy)-N-(4-(vinylsulfonyl)phenyl)-9H-purin-2-amine

References

1. Anscombe E, et al. Chem Biol. 2015 Sep 17;22(9):1159-64.

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NU-6300 (NU 6300;NU6300)

Biological Activity

Physicochemical Properties

References

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