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Chemical Structure : PSB-KD107
Catalog No.: PC-49030Not For Human Use, Lab Use Only.
PSB-KD107 is a potent, selective GPR18 receptor agonist with EC50 of 0.562 uM and 1.78 uM for human and mouse GPR18, respectively.
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PSB-KD107 is a potent, selective GPR18 receptor agonist with EC50 of 0.562 uM and 1.78 uM for human and mouse GPR18, respectively.
PSB-KD107 produces concentration-dependent relaxation in phenylephrine-precontracted endothelium-intact aortic rings with pIC50 of 5.22.
PSB-KD107 exerts vascular activity and produces total relaxation of phenylephrine-pre-contracted rat aorta.
| M.Wt | 378.436 | |
| Formula | C20H22N6O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Magdalena Kotańska, et al. Pharmaceuticals (Basel). 2021 Aug 13;14(8):799.
2. Andhika B Mahardhika, et al. J Med Chem. 2024 Jun 17. doi: 10.1021/acs.jmedchem.3c02423.
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