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SR-16430

Chemical Structure : SR-16430

CAS No.: 612837-86-2

SR-16430 (SR16430)

Catalog No.: PC-61538Not For Human Use, Lab Use Only.

SR-16430 is a selective ORL1 receptor (NOP receptor) antagonist that has 10-fold selectivity over μ-opioid receptor.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    SR-16430 is a selective ORL1 receptor (NOP receptor) antagonist that has 10-fold selectivity over μ-opioid receptor.

    Physicochemical Properties

    M.Wt 369.472
    Formula C21H30F3NO
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    1-(cyclooctylmethyl)-4-(3-(trifluoromethyl)phenyl)piperidin-4-ol

    References

    1. Khroyan TV, et al. J Pharmacol Exp Ther. 2007 Feb;320(2):934-43.

    2. Spagnolo B, et al. Br J Pharmacol. 2008 Feb;153(3):609-19.

    3. Khroyan TV, et al. Eur J Pharmacol. 2009 May 21;610(1-3):49-54.

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