Chemical Structure : Vorapaxar
CAS No.:
618385-01-6
Vorapaxar
(SCH530348, SCH-530348, SCH 530348)
Catalog No. : PC-42330Not For Human Use, Lab Use Only.
Vorapaxar (SCH 530348) is a potent, selective and orally active thrombin receptor PAR-1 antagonist with Ki of 8.1 nM.
Packing Price Stock Quantity 5 mg $88 In stock 0 1 2 3 4 5 10 mg $128 In stock 0 1 2 3 4 5 25 mg $218 In stock 0 1 2 3 4 5 50 mg $358 In stock 0 1 2 3 4 5 100 mg $558 In stock 0 1 2 3 4 5 250 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4233001
Biological Activity
Vorapaxar (SCH 530348) is a potent, selective and orally active thrombin receptor PAR-1 antagonist with Ki of 8.1 nM.
Physicochemical Properties
M.Wt
492.5817
Formula
C29H33FN2O4
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 30 mg/mL
Chemical Name/SMILES
Carbamic acid, N-[(1R,3aR,4aR,6R,8aR,9S,9aS)-9-[(1E)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]dodecahydro-1-methyl-3-oxonaphtho[2,3-c]furan-6-yl]-, ethyl ester
References
1. Chackalamannil S, et al. J Med Chem.
2. Chintala M, et al. J Pharmacol Sci.
3. Goto S, et al. J Atheroscler Thromb
4. Becker RC, et al. Lancet.
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