eN-IN-1 |CAS:95523-13-0 Probechem Biochemicals

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Chemical Structure : eN-IN-1

eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine)

Catalog No.: PC-42064Not For Human Use, Lab Use Only.

An α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 29 nM for rat recombinant eN.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine) is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 29 nM for rat recombinant eN.
eN-IN-1 also exhibits dual-action properties toward both A2AR and equilibrative nucleoside transporter 1 (ENT1) with Ki of 27.7 uM and 6.51 nM.

Physicochemical Properties

M.Wt	372.3785
Formula	C17H20N6O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Adenosine, N-[(4-aminophenyl)methyl]-

References

1. Bhattarai S, et al. J Med Chem. 2015 Aug 13;58(15):6248-63.

2. Chen JB, et al. ChemMedChem. 2011 Aug 1;6(8):1390-400.

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eN-IN-1 (N-[(4-Aminophenyl)methyl]adenosine)

Biological Activity

Physicochemical Properties

References

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