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Chemical Structure : hM3Dq-agonist-21
CAS No.: 56296-18-5
Catalog No.: PC-42096Not For Human Use, Lab Use Only.
hM3Dq-agonist-21 is a potent, selective human muscarinic acetylcholine M3 receptor (hM3Dq) full agonist with EC50 of 1.7 nM.
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|---|---|---|---|
| 10 mg | $128 | In stock | |
| 25 mg | $198 | In stock | |
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| 100 mg | Get quote |
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hM3Dq-agonist-21 is a potent, selective human muscarinic acetylcholine M3 receptor (hM3Dq) full agonist with EC50 of 1.7 nM.
hM3Dq-agonist-21 displays 3.5-fold selective over H1, 40-fold selective over 5HT2A, 100-fold selective over 5HT2C, 165-fold selective over α1A, and inactive at native human M3 receptor (hM3).
| M.Wt | 278.3516 | |
| Formula | C17H18N4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 78 mg/mL |
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| Chemical Name/SMILES |
5H-Dibenzo[b,e][1,4]diazepine, 11-(1-piperazinyl)- |
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1. Chen X, et al. ACS Chem Neurosci. 2015 Mar 18;6(3):476-84.
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