CRF Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-25856	CRF1 Receptor Antagonist M43 CRF1 antagonist	CRF1 Receptor Antagonist M43 is a potent, selective nonpeptide corticotropin-releasing factor receptor 1 (CRHR1, CRF1) with Ki of 19.2 nM.
PC-25842	Antalarmin hydrochloride CRF1 antagonist	Antalarmin hydrochloride is a potent, selective nonpeptide corticotropin-releasing factor receptor 1 (CRHR1, CRF1) antagonist with Ki of 2.7 nM, with no effect on CRF2 receptor.
PC-21400	K41498 CRF2 inhibitor	K41498 is a potent, highly selective CRF2 receptor antagonist with Ki values of 0.66 nM, 0.62 nM and 425 nM for human CRF2α, CRF2β and CRF1 receptors respectively.
PC-21399	NBI-35965 CRF1 inhibitor	NBI-35965 is a potent, selective antagonist of corticotropin-releasing factor 1 (CRF1) receptor with Ki of 4 nM, >1000-fold selective over CRF2.
PC-21195	BMK-C205 CRF1R inhibitor	BMK-C205 (BMK-C 205) is a potent, selective corticotropin-releasing hormone receptor 1 (CRF1R) antagonist with IC50 of 74 nM in calcium mobilization assays, blocks hypothalamus-pituitary-adrenal (HPA) axis activation.

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