Cat. No. |
Product Name |
Information |
PC-60270 |
G-1
|
GPER/GPR30 agonist G-1 (Tespria) is potent and selective GPER/GPR30 agonist with Ki of 11 nM, EC50 of 2 nM. |
PC-60268 |
G-15
|
G-15 (GPR30 inhibitor G15, G15) is a potent, selective GPER/GPR30 antagonist with Ki of 20 nM. |
PC-60269 |
G-36
|
A potent, selective, cell-permeable GPER/GPR30 antagonist that inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 with IC50 of 112 nM and 165 nM, respectively. |