| Cat. No. |
Product Name |
Information |
| PC-72357 |
GPR84 antagonist 837
GPR84 antagonist
|
Compound 837 (GPR84 antagonist) is a highly potent (affinity, 1 nM), selective antagonist of both orthosteric and allosteric activators of GPR84. |
| PC-72356 |
GLPG1205
GPR84 antagonist
|
GLPG1205 is a potent and selective GPR84 inhibitor (negative allosteric modulator) with IC50 of 54 nM (hGPR84). |
| PC-43189 |
6-OAU
GPR84 agonist
|
6-OAU (GTPL5846, 6-n-Octylaminouracil) is a potent, specific agonist of GPR84 with EC50 of 512 nM in [35S]GTPγS binding assay, without activity for GPR109A and OXER1 in a panel of 69 GPCRs. |