| Cat. No. |
Product Name |
Information |
| PC-24434 |
TUG-2099
GPR84 agonist
|
TUG-2099 is a potent, selective GPR84 agonist with EC50 of 0.3 nM (hGPR84), Emax=84%. |
| PC-24433 |
TUG-2181
GPR84 antagonist
|
TUG-2181 is a potent, selective antagonist of GPR84 with pIC50 of 7.66 and 5.89 for hGPR84 and mGPR84 respecitvely in cAMP assays. |
| PC-21649 |
PSB-16434
GPR84 agonist
|
PSB-16434 is a highly potent, Gi pathway-selective GPR84 agonist with cAMP EC50 of 7.1 nM, 79-fold selective over β-arrestin-2 recruitment activity. |